CAS NO: | 2361114-15-8 |
包装: | 50mg, 100mg, 250mg |
规格: | ≥98% |
PROTAC ER Degrader-4 is a PROATC estrogen receptor (ER) degrader, binding to ER with an IC50 of 0.8 nM. PROTAC ER Degrader-4 induces ER degradation in MCF-7 cells with an IC50 of 0.3 nM. References: [1]. Bin Yang, et al. Compounds and their use in treating cancer. WO2019123367A1.
纯度:≥98%
CAS:2361114-15-8